Stephania Fa Cepharanthine Powder

Orukọ ọja: Stephania Japonica Extract
Orisun Latin: Stephania cephalantha Hayata(Stephania japonica (Thunb.) Miers)/ Stephania epigaea Lo/ Stephania yunnanensis HSLo.
Irisi: funfun, grẹy White Powder
Eroja ti nṣiṣe lọwọ: Cepharanthine 80% -99% HPLC
Apakan Lo: Tuber/Root
Ohun elo: Awọn ọja ilera
Ojutu yo: 145-155°
Yiyi ni pato: D20+277°(c=2inchloroform)
Ojutu farabale: 654.03°C (iṣiro ti o ni inira)
iwuwo: 1.1761 (iṣiro ti o ni inira)
Atọka itọka: 1.5300 (iṣiro)
Awọn ipo ipamọ: underinertgas (nitrogen tabi Argon) ni 2-8 ° C
Solubility: Soluble ni SO (35mg/ml) tabi ethanol (20mg/ml)
Olusọdipúpọ acidity (pKa): 7.61 ± 0.20 (Asọtẹlẹ)


Alaye ọja

Awọn alaye miiran

ọja Tags

Ọja Ifihan

Stephania Extract Cepharanthine Powder jẹ nkan ti o wa lati awọn isu ti ọgbin Stephania cephalantha Hayata (Stephania japonica (Thunb.) Miers) tabi Stephania epigaea Lo/ Stephania yunnanensis HSLo.Cepharanthine jẹ ọja adayeba ti o ya sọtọ lati inu ọgbin yii ati pe o ti jẹ koko-ọrọ ti ọpọlọpọ awọn ijinlẹ nitori awọn ohun-ini elegbogi ti o pọju.O ti rii lati ṣafihan awọn iṣẹ egboogi-SARS-CoV-2, ti n ṣafihan imunadoko ni didapa itankale ọlọjẹ.Ni afikun, Cepharanthine ti ṣe afihan agbara lati yiyipada P-glycoprotein (P-gp) -aabo idawọle olopobobo ninu awọn sẹẹli kan ati mu ifamọ ti awọn aṣoju anticancer ni awọn awoṣe idanwo.Pẹlupẹlu, o ti han lati ni awọn ipa ti o ni idiwọ lori ẹdọ cytochrome P450 awọn enzymu CYP3A4, CYP2E1, ati CYP2C9, ati pe o ni nkan ṣe pẹlu antitumor, egboogi-iredodo, ati awọn ipa antinociceptive.
Ni akojọpọ, Stephania Extract Cepharanthine Powder jẹ fọọmu ti o ni erupẹ ti ọja adayeba Cepharanthine ti o wa lati inu ọgbin Stephania cephalantha, eyiti o ti ṣe afihan agbara ni orisirisi awọn ohun elo oogun.

Sipesifikesonu (COA)

Ọja Cepharanthine
CAS 481-49-2
Ayẹwo 80% ~ 99%
Ifarahan funfun lulú
Iṣakojọpọ 1KG/Apo bankanje
Nkan Sipesifikesonu
Ifarahan grẹy funfun lulú, didoju wònyí, gíga hygroscopic
Idanimọ TLC: Ojutu boṣewa ati ojutu idanwo aaye kanna, RF
Ayẹwo (Ipilẹ gbigbẹ) 98.0% --102.0%
Specific Optical -2.4°~ -2.8°
PH 4.5 ~ 7.0
Awọn irin Heavy (Bi Pb) ≤10ppm
As ≤1ppm
Pb ≤0.5ppm
Cd ≤1ppm
Hg ≤0.1pm
Ohun elo ti o jọmọ Aami ko tobi ju aaye ojutu boṣewa lọ
Aloku to ku <0.5%
Omi akoonu <2%

Ọja Awọn ẹya ara ẹrọ

Stephania Extract Cepharanthine Powder jẹ ọja adayeba ti o wa lati inu ọgbin Stephania cephalantha Hayata.O ti rii pe o ni ọpọlọpọ awọn ohun-ini elegbogi, pẹlu:
1. Anti-SARS-CoV-2 akitiyan
2. Awọn ipa idinamọ lori ilọsiwaju ti gbogun ti
3. Iyipada ti P-glycoprotein-mediated multidrug resistance
4. Imudara ifamọ si awọn aṣoju anticancer
5. Awọn ipa idiwọ lori ẹdọ cytochrome P450 awọn enzymu CYP3A4, CYP2E1, ati CYP2C9
6. Antitumor, egboogi-iredodo, ati awọn ipa antinociceptive

Kini Biosynthesis ti Cepharanthine?

Biosynthesis ti cepharanthine ni Stephania bẹrẹ pẹlu ifasilẹ ti dopamine ati 4-hydroxyphenylacetaldehyde (4-HPAA, 5) nipasẹ norcoclaurine synthase (NCS), ti nso norcoclaurine.

Kini Solubility ti Cepharanthine?

Cepharanthine jẹ tiotuka ninu awọn nkan ti o ni nkan ti ara ẹni gẹgẹbi ethanol, DMSO, ati dimethyl formamide (DMF).Solubility ti cepharanthine ninu awọn olomi wọnyi jẹ isunmọ 2, 5, ati 10 mg/ml, lẹsẹsẹ.Cepharanthine jẹ tiotuka diẹ ninu awọn buffer olomi.

Awọn ohun elo

Awọn ile-iṣẹ ohun elo fun Stephania Extract Cepharanthine Powder pẹlu Pharmaceutical, Nutraceutical, Biotechnology, and Herbal Medicine, awọn ohun elo akọkọ jẹ bi atẹle:
O pọju lilo ni antiviral awọn itọju ailera
O pọju bi oluranlọwọ ni itọju akàn
O pọju fun lilo ninu awọn itọju egboogi-iredodo
O pọju bi oluranlowo analgesic
Awọn ohun elo wọnyi ṣe afihan awọn lilo agbara oniruuru ti Stephania Extract Cepharanthine Powder ni orisirisi awọn ipo itọju ailera.


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